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Macrocycles in new drug discovery | Future Medicinal Chemistry
Macrocycles in new drug discovery | Future Medicinal Chemistry

Direct small-molecule inhibitors of KRAS: from structural insights to  mechanism-based design | Nature Reviews Drug Discovery
Direct small-molecule inhibitors of KRAS: from structural insights to mechanism-based design | Nature Reviews Drug Discovery

DNA-encoded chemistry: enabling the deeper sampling of chemical space |  Nature Reviews Drug Discovery
DNA-encoded chemistry: enabling the deeper sampling of chemical space | Nature Reviews Drug Discovery

Mechanistic enzymology in drug discovery: a fresh perspective | Nature  Reviews Drug Discovery
Mechanistic enzymology in drug discovery: a fresh perspective | Nature Reviews Drug Discovery

The drug–target residence time model: a 10-year retrospective | Nature  Reviews Drug Discovery
The drug–target residence time model: a 10-year retrospective | Nature Reviews Drug Discovery

Investigating antimalarial drug interactions of emetine dihydrochloride  hydrate using CalcuSyn-based interactivity calculations
Investigating antimalarial drug interactions of emetine dihydrochloride hydrate using CalcuSyn-based interactivity calculations

Biophysics in drug discovery: impact, challenges and opportunities | Nature  Reviews Drug Discovery
Biophysics in drug discovery: impact, challenges and opportunities | Nature Reviews Drug Discovery

Contribution of NIH funding to new drug approvals 2010–2016 | PNAS
Contribution of NIH funding to new drug approvals 2010–2016 | PNAS

Covalent fragment libraries in drug discovery - ScienceDirect
Covalent fragment libraries in drug discovery - ScienceDirect

Screening-based approach to discover effective platinum-based  chemotherapies for cancers with poor prognosis
Screening-based approach to discover effective platinum-based chemotherapies for cancers with poor prognosis

Drug design from the cryptic inhibitor envelope | Nature Communications
Drug design from the cryptic inhibitor envelope | Nature Communications

Creating and screening natural product libraries - Natural Product Reports  (RSC Publishing) DOI:10.1039/C9NP00068B
Creating and screening natural product libraries - Natural Product Reports (RSC Publishing) DOI:10.1039/C9NP00068B

The drug–target residence time model: a 10-year retrospective | Nature  Reviews Drug Discovery
The drug–target residence time model: a 10-year retrospective | Nature Reviews Drug Discovery

CISNE: An accurate description of dose-effect and synergism in combination  therapies | Scientific Reports
CISNE: An accurate description of dose-effect and synergism in combination therapies | Scientific Reports

A Comprehensive Biophysical Analysis of the Effect of DNA Binding Drugs on  Protamine-induced DNA Condensation | Scientific Reports
A Comprehensive Biophysical Analysis of the Effect of DNA Binding Drugs on Protamine-induced DNA Condensation | Scientific Reports

DeepConv-DTI: Prediction of drug-target interactions via deep learning with  convolution on protein sequences
DeepConv-DTI: Prediction of drug-target interactions via deep learning with convolution on protein sequences

Organ‐on‐chip models: Implications in drug discovery and clinical  applications - Mittal - 2019 - Journal of Cellular Physiology - Wiley  Online Library
Organ‐on‐chip models: Implications in drug discovery and clinical applications - Mittal - 2019 - Journal of Cellular Physiology - Wiley Online Library

Computational design of substrate selective inhibition
Computational design of substrate selective inhibition

Drug development - Wikipedia
Drug development - Wikipedia

Covalent fragment libraries in drug discovery - ScienceDirect
Covalent fragment libraries in drug discovery - ScienceDirect

PDF) Metal–ligand interactions in drug design
PDF) Metal–ligand interactions in drug design

IJMS | Free Full-Text | Key Topics in Molecular Docking for Drug Design |  HTML
IJMS | Free Full-Text | Key Topics in Molecular Docking for Drug Design | HTML

PDF) The nature of ligand efficiency
PDF) The nature of ligand efficiency